{"product_id":"retatrutide","title":"Retatrutide","description":"\u003ch4\u003e\u003cspan class=\"\"\u003eAbout the Product\u003c\/span\u003e\u003c\/h4\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eGenetic Labs Retatrutide\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e is a high-purity synthetic peptide (research grade) supplied in a vial containing 20mg of lyophilized (freeze-dried) powder. Retatrutide is a novel, tri-agonist peptide that simultaneously targets three key metabolic hormone receptors: the \u003c\/span\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eglucagon-like peptide-1 receptor (GLP-1R)\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e , the \u003c\/span\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eglucose-dependent insulinotropic polypeptide receptor (GIPR)\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e , and the \u003c\/span\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eglucagon receptor (GCGR)\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e . This unique triple agonism represents a significant advancement in metabolic research, offering a multi-pathway approach to studying energy balance, glucose homeostasis, and lipid metabolism.\u003c\/span\u003e\u003c\/p\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eKit Contents:\u003c\/span\u003e\u003c\/strong\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cspan class=\"\"\u003e1 Vial with 20mg Retatrutide (Lyophilized Powder)\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cspan class=\"\"\u003e1 Vial with 3mL Bacteriostatic Water (Diluent)\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eFor Laboratory Research Use Only. Not for human consumption.\u003c\/span\u003e\u003c\/strong\u003e\u003c\/p\u003e\n\u003chr\u003e\n\u003ch4\u003e\u003cspan class=\"\"\u003eBenefits (Research Scope)\u003c\/span\u003e\u003c\/h4\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eTriple Receptor Agonist:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Retatrutide is the first-in-class peptide that activates all three receptors—GLP-1R, GIPR, and GCGR—simultaneously. This unique combination allows researchers to study the synergistic effects of multiple metabolic pathways in a single compound, offering advantages over selective or dual agonists.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eVersatile Research Tool:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Suitable for a wide range of studies, including:\u003c\/span\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eMetabolic Disorders:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Research into obesity, type 2 diabetes, metabolic syndrome, and non-alcoholic fatty liver disease (NAFLD).\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eEnergy Expenditure:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Studies on resting energy expenditure, thermogenesis, and brown adipose tissue (BAT) activation.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eLipid Metabolism:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Research into fatty acid oxidation, lipolysis, and lipid profiling.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eAppetite \u0026amp; Body Weight:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Studies on hypothalamic regulation of food intake, satiety, and sustained weight reduction.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eGlucose Homeostasis:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Investigation into insulin secretion, glucagon regulation, and glycemic control.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eCardiovascular Research:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Studies on cardiovascular outcomes, blood pressure, and lipid profiles.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003ePractical Formulation:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e The lyophilized powder ensures stability and extended shelf life, while the included bacteriostatic water facilitates easy reconstitution for both \u003c\/span\u003e\u003cem\u003e\u003cspan class=\"\"\u003ein vitro\u003c\/span\u003e\u003c\/em\u003e\u003cspan class=\"\"\u003e and \u003c\/span\u003e\u003cem\u003e\u003cspan class=\"\"\u003ein vivo\u003c\/span\u003e\u003c\/em\u003e\u003cspan class=\"\"\u003e experiments.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003chr\u003e\n\u003ch4\u003e\u003cspan class=\"\"\u003eResearch \u0026amp; Science\u003c\/span\u003e\u003c\/h4\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cspan class=\"\"\u003eRetatrutide is a groundbreaking investigational peptide that has generated significant interest in the scientific community for its multi-targeted approach to metabolic disease research.\u003c\/span\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eMechanism of Action:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Retatrutide is a 39-amino-acid peptide engineered to bind and activate three distinct receptors:\u003c\/span\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eGLP-1R (Glucagon-Like Peptide-1 Receptor):\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Stimulates glucose-dependent insulin secretion, suppresses glucagon, slows gastric emptying, and reduces appetite.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eGIPR (Glucose-Dependent Insulinotropic Polypeptide Receptor):\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Enhances insulin secretion, improves lipid metabolism, and reduces adiposity.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eGCGR (Glucagon Receptor):\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Increases energy expenditure, stimulates lipolysis, promotes fatty acid oxidation, and enhances thermogenesis.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eTriple Agonism Advantage:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e The combination of these three pathways results in a coordinated metabolic effect that goes beyond the capabilities of GLP-1 agonists alone:\u003c\/span\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eGLP-1R + GIPR:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Enhanced insulin secretion, improved glycemic control, and synergistic weight loss effects.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eGIPR + GCGR:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Amplified lipid metabolism and energy expenditure.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eGLP-1R + GCGR:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Optimized glucose homeostasis with balanced energy utilization.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003ePreclinical Research:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Studies have demonstrated that retatrutide:\u003c\/span\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eSignificantly reduces body weight\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e and adiposity in diet-induced obesity models, with greater efficacy than GLP-1R or GIPR selective agonists.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eImproves glycemic control\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e with superior glucose-lowering effects compared to semaglutide.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eEnhances lipid metabolism\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e with reductions in triglycerides, LDL cholesterol, and hepatic steatosis.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eIncreases energy expenditure\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e through activation of brown adipose tissue (BAT) and increased thermogenesis.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eClinical Research:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Retatrutide has been evaluated in clinical trials, including dose-escalation studies in individuals with obesity and type 2 diabetes, demonstrating:\u003c\/span\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cspan class=\"\"\u003eSubstantial weight loss (up to 24% reduction in body weight in clinical trials).\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cspan class=\"\"\u003eSignificant improvements in glycemic control and HbA1c reduction.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cspan class=\"\"\u003eFavorable cardiovascular and renal outcome profiles.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cspan class=\"\"\u003eThe unique triple agonist mechanism may contribute to greater metabolic benefits compared to current GLP-1-based therapies.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eNeuroprotective Research:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Emerging research is exploring retatrutide's potential in neurodegenerative diseases, as GLP-1R and GIPR are expressed in the brain, and their activation has been shown to reduce neuroinflammation and improve cognitive function.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003eFocus on Genetic Variability:\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e Current research is investigating how genetic polymorphisms in GLP1R, GIPR, GCGR, and other metabolic pathway genes may influence individual responses to retatrutide, providing insights for personalized metabolic interventions.\u003c\/span\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e\n\u003chr\u003e\n\u003ch3\u003e\u003cspan class=\"\"\u003eImportant Note on Kit Contents\u003c\/span\u003e\u003c\/h3\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cspan class=\"\"\u003ePlease verify the kit contents as listed in the image:\u003c\/span\u003e\u003c\/p\u003e\n\u003cul\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003e1 x Vial Retatrutide (Lyophilized Powder) 20mg\u003c\/span\u003e\u003c\/strong\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003cli\u003e\n\u003cp class=\"ds-markdown-paragraph\"\u003e\u003cstrong\u003e\u003cspan class=\"\"\u003e1 x Vial Bacteriostatic Water (Diluent) 3mL\u003c\/span\u003e\u003c\/strong\u003e\u003cspan class=\"\"\u003e \u003c\/span\u003e\u003cem\u003e\u003cspan class=\"\"\u003e(Note: The text in the image appears to have a typo. It should read \"Bacteriostatic Water\" as per standard practice.)\u003c\/span\u003e\u003c\/em\u003e\u003c\/p\u003e\n\u003c\/li\u003e\n\u003c\/ul\u003e","brand":"Genetic Labs","offers":[{"title":"5mg","offer_id":58672597369157,"sku":null,"price":78.0,"currency_code":"EUR","in_stock":true},{"title":"20mg","offer_id":58672597401925,"sku":null,"price":178.0,"currency_code":"EUR","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/1077\/7614\/7781\/files\/GeneticLabs-Retatrutide_5mg.jpg?v=1784937315","url":"https:\/\/genetic-peps.shop\/products\/retatrutide","provider":"Genetic Peps","version":"1.0","type":"link"}